PT-141 (nasal spray) 100 mg/ml (5ml)

$239.00

Delivery T&C

PT-141 (bremelanotide) is a melanocortin (MC3R/MC4R) receptor agonist that acts on central nervous system pathways and is available only by prescription when a licensed healthcare provider determines it is clinically appropriate for an individual patient.

Not Available in: AL, AR, IN, MN

Unlike Viagra or Cialis which only improve blood flow, PT-141 boosts libido and sexual motivation at the neurological level — making it a commonly discussed option for those who want to support sexual drive, sensitivity, and intimacy. Your provider will evaluate whether PT-141 is appropriate for your situation.

  • Unique melanocortin receptor agonist that works in the brains’ arousal centers
  • Available as injection (10mg/ml) or nasal spray for convenience
  • Non-hormonal approach to sexual vitality and libido health for both men and women
  • Can produce erections even without visual stimulation; enhances rigidity and duration in studies
  • Fast-acting with on-demand potential; 30-60min potential
PT-141 (bremelanotide) is the active ingredient in FDA-approved Vyleesi (injection, for HSDD in premenopausal women). This compounded nasal spray is not FDA-approved, is not Vyleesi, and is not reviewed by the FDA for safety, effectiveness, or quality. Any use is at a licensed provider’s independent clinical discretion; where prescribed, it is compounded by a state-licensed 503A pharmacy under a patient-specific prescription and shipped to the patient. Defy Age RX does not dispense medication; no product is provided without a valid prescription. Individual results vary. Not medical advice.
  • Increased sexual desire and arousal in men and women
  • Improved performance, stamina, and satisfaction
  • Enhanced sensitivity and pleasure
  • Works independently of vascular mechanisms (unlike PDE5 inhibitors,Viagra)
AspectSubcutaneous InjectionNasal Spray
Bioavailability & ConsistencyHigher and more predictable (stable plasma levels)Lower and more variable (affected by congestion, technique, allergies)
Onset~30–60 minutes (often ~45 min)~20–60 minutes (potentially slightly faster brain access)
DurationOften 6–12 hours (duration may vary by individual)Typically 4–6 hours (sometimes shorter)
Potency & EffectivenessGenerally stronger, more reliable results; better for moderate-severe cases or inconsistent respondersEffective for mild cases; good but less consistent magnitude
Ease of UseRequires self-injection (small needle, abdomen/thigh); quick once comfortableNeedle-free, highly convenient and discreet
DosingStandard: 1.75 mg (FDA-approved Vyleesi for women; off-label similar for men)Often 0.5–1 mg (or higher in compounded forms); variable absorption
Side EffectsSimilar profile; possible injection-site reactions (redness, pain)Similar (nausea ~40%, flushing, headache); sometimes fewer systemic effects at lower doses; nasal irritation possible
Best ForMaximum reliability, stronger effects, longer durationConvenience, needle aversion, discretion, maintenance or mild needs

PT-141, Tadalafil, CJC-1295 – a combination sometimes discussed in clinical contexts. Read Full Article

PT-141 and BPC-157

 

PT-141 and Tadalafil – a commonly paired combination for sexual health. Your provider will evaluate appropriateness for your individual situation.

 

Prescribed after telehealth consultation and shipped discreetly from our partner 503A pharmacy. Room-temperature or mild refrigeration shipping. Most orders fulfilled within 4–8 business days.
This product is compounded and not FDA-approved. It has not been evaluated by the FDA for safety, efficacy, or quality. It requires a valid prescription following a medical consultation with a licensed healthcare provider. Individual results may vary and are not guaranteed. Not intended to diagnose, treat, cure, or prevent any disease. Results depend on lifestyle factors and this product is not a substitute for medical care.

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A note about FDA compliance: *The doctor network may prescribe certain compounded drugs for the treatment of certain conditions,
subject to approval by a provider through the DefyAgeRX; however, even though our partner pharmacies use only pharmaceutical-grade
ingredients and are highly regulated, compounded prescriptions are not FDA approved. The appearance, contents, and dosage of the vial
may vary based on your personalized prescription, and individual results may vary.

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